Título : New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models |
Autor : Fernandez-Carvajal, Asia  Di Sarno, Veronica Giovannelli, Pia  Medina Peris, Alicia  Ciaglia, Tania Di Donato, Marzia Musella, Simona  Lauro, Gianluigi  Vestuto, Vincenzo  Smaldone, Gerardina  Di Matteo, Francesca BIFULCO, Giuseppe  Castoria, Gabriella  Migliaccio, Antimo  Campiglia, Pietro  Gomez Monterrey, Isabel Maria  Ostacolo, Carmine BERTAMINO, Alessia  |
Editor : Elsevier |
Departamento: Departamentos de la UMH::Bioquímica y Biología Molecular |
Fecha de publicación: 2022 |
URI : https://hdl.handle.net/11000/34384 |
Resumen :
TRPM8 has recently emerged as a druggable target in prostate cancer (PC) and TRPM8 modulators have been
proposed as potential anticancer agents in this pathology. We have recently demonstrated their effectiveness in a castration-resistant prostate cancer (CRPC) model that is usually resistant to an... Ver más
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Palabras clave/Materias: TRPM8 antagonists Ca2+-microfluorimetric assays Electrophysiology Anticancer activity Castration-resistant prostate cancer cells Spheroids |
Área de conocimiento : CDU: Ciencias puras y naturales: Biología: Bioquímica. Biología molecular. Biofísica |
Tipo de documento : info:eu-repo/semantics/article |
Derechos de acceso: info:eu-repo/semantics/closedAccess Attribution-NonCommercial-NoDerivatives 4.0 Internacional |
DOI : https://doi.org/10.1016/j.ejmech.2022.114435 |
Publicado en: European Journal of Medicinal Chemistry |
Aparece en las colecciones: Artículos Bioquímica y Biología Molecular
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