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2021_02_Nikolaeva_Scientific reports_2021_AG1529.pdf.jpgJan-2021A capsaicinoid‑based soft drug, AG1529, for attenuating TRPV1‑mediated histaminergic and infammatory sensory neuron excitability
Nikolaeva Koleva, Magdalena; Butron, Laura; González-Rodríguez, Sara; Devesa Giner, Isabel; Valente, Pierluigi; Serafni, Marta
1- Journal of Medicinal Chemistry 2020.pdf.jpg2020Exploration of TRPM8 Binding Sites by β‑Carboline-Based Antagonists and Their In Vitro Characterization and In Vivo Analgesic Activities
Fernandez-Carvajal, Asia; BERTAMINO, Alessia; Ostacolo, Carmine; Medina Peris, Alicia; Di Sarno, Veronica; Lauro, Gianluigi; Ciaglia, Tania; Vestuto, Vincenzo; Di Giacomo Pepe , Giuseppe; Basilicata, Manuela Giovanna; Musella, Simona; Smaldone, Gerardina; Cristiano, Claudia; González-Rodríguez, Sara; Bifulco, Giuseppe; Campiglia, Pietro; Gomez Monterrey, Isabel Maria; Russo, Roberto
s41598-020-70691-x.pdf.jpg2020Highly functionalized β‑lactams and 2‑ketopiperazines as TRPM8 antagonists with antiallodynic activity
Bonache, M. Ángeles; Martín Escura, Cristina; De la Torre Martínez, Roberto; Medina, Alicia; González-Rodríguez, Sara; Francesch, Andres; Cuevas, Carmen; Roa, Ana María; Fernández-Ballester, Gregorio; Ferrer-Montiel, Antonio; Fernández Carvajal, Asia; González-Muñiz, Rosario